Hexarelin – Aliquot, 5mg

$44.99

Hexarelin – Aliquot, 5mg is ultra-pure, analytical-grade synthetic growth hormone secretagogue (GHS) peptide with 99% purity, designed for in vitro/in vivo endocrine research and analytical testing. This lyophilized material functions as a potent ghrelin receptor (GHS-R1a) agonist and one of the most potent stimulators of growth hormone (GH) release available in the GHS class, releasing GH from pituitary somatotrophs in a dose-dependent manner and increasing insulin-like growth factor 1 (IGF-1) secretion, with a 6-amino acid sequence (His-D-2-Me-Trp-Ala-Trp-D-Phe-Lys-NH₂), making it invaluable for investigators studying GH-axis biology, anti-aging research, muscle growth mechanisms, fat metabolism, recovery enhancement, neuroendocrine regulation, and CD36 receptor signaling pathways. Hexarelin retains efficacy even in the presence of somatostatin inhibition, though it induces rapid receptor desensitization (tachyphylaxis) in long-term models. Available for fast, compliant shipping to all U.S. states and European countries via dedicated logistics hubs.

  • Third-party certified lot coding with publicly available COA (Certificate of Analysis) for absolute purity transparency

  • Formulation completely free of adulterants, excipients, flow agents, and other compounds to guarantee raw chemical purity

  • Precision over-weighed by 5-10% inside vessel to compensate for natural adhesion loss during laboratory powder transfer

  • UV-resistant lyophilized vial with tamper-proof seal engineered for transit safety and chemical stability

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Description

Hexarelin – Aliquot, 5mg

This premium, laboratory-grade research compound delivers ultra-pure synthetic Hexarelin peptide at 99% purity, representing the highest standard for modern scientific investigations into growth hormone secretagogue-mediated GH secretion and IGF-1 augmentation mechanisms. The lyophilized aliquot format provides investigators with a ready-to-reconstitute single-compound reference standard ideal for analytical testing, in vitro pituitary cell culture modeling, and in vivo preclinical research applications where precise Hexarelin administration is critical for studying potent GH release dynamics, ghrelin receptor activation, and neuroendocrine regulation.

All shipments to the 50 United States are fulfilled directly from primary U.S. production facilities, ensuring 2-5 business day delivery nationwide. International orders to the United Kingdom and continental Europe are processed through our dedicated United Kingdom shipping hub, which streamlines customs clearance and reduces transit times across all European countries. This dual-hub logistics infrastructure guarantees seamless, compliant delivery while maintaining peptide integrity throughout transit.

  • Public third-party lab reports with unique lot-coding ensure absolute transparency for every batch sold

  • Formulation contains zero adulterants, excipients, flow agents, or contaminants—pure Hexarelin peptide only

  • Strategic over-packaging compensates for peptide adhesion loss, guaranteeing minimum 5mg recoverable material

  • Lyophilized vial features UV-resistant construction and tamper-proof seal for transit safety


Technical Specifications & Chemical Profile

Chemical Property Specification Data
Product Name Hexarelin – Aliquot, 5mg
Common Synonyms Hexarelin Acetate, Examorelin, GHRP-6 Analogue, Growth Hormone-Releasing Peptide-6 Analogue, GHS Agonist
CAS Number 140703-51-1
Molecular Formula C₄₇H₅₈N₁₂O₆
Molar Mass 887.04 g/mol
Primary Target Mechanism Synthetic hexapeptide; growth hormone secretagogue (GHS); ghrelin receptor (GHS-R1a) agonist; potent GH secretagogue active after two successive doses; dose-dependent GH release from pituitary somatotrophs; increases IGF-1 secretion; 6-amino acid sequence (His-D-2-Me-Trp-Ala-Trp-D-Phe-Lys-NH₂); chemically modified from GHRP-6 to enhance stability and potency via D-2-Me-Trp² substitution; retains efficacy in presence of somatostatin (SRIF) inhibition; synergistic with GHRH (Growth Hormone-Releasing Hormone); loses synergistic property after repeated administration; rapid receptor desensitization (tachyphylaxis) in long-term models; potentially acts via CD36 receptor; stimulates muscle growth; improves recovery; aids fat loss; anti-aging effects; neuroendocrine regulation; half-life: short (minutes); potent GH release; no increase of appetite
Physical Form Lyophilized white to off-white powder (aliquot vial)

Research Applications & Storage Protocols

GHS-R1a Agonism & Potent GH/IGF-1 Secretion Profiling

Hexarelin (Hexarelin Acetate, Examorelin) functions as a synthetic hexapeptide belonging to the Growth Hormone Secretagogue (GHS) family, structurally related to GHRP-6 but chemically modified to enhance stability and potency through the D-2-Me-Trp² substitution in its sequence. The compound is a 6-amino acid peptide with the sequence His-D-2-Me-Trp-Ala-Trp-D-Phe-Lys-NH₂, making it one of the most potent stimulators of Growth Hormone release available in the GHS class. Preclinical research identifies Hexarelin as acting via the Ghrelin receptor (GHS-R1a) and potentially the CD36 receptor, releasing growth hormone from the pituitary gland in a dose-dependent manner. Unlike other secretagogues, studies suggest Hexarelin retains efficacy even in the presence of somatostatin (SRIF) inhibition, demonstrating unique resistance to this native GH-inhibiting hormone. Hexarelin and GHRH (Growth Hormone-Releasing Hormone) are synergistic, a property which is lost after repeated administration, and the compound is a potent GH secretagogue active after two successive doses, with the magnitude of the GH response to the second dose influenced by the dosing interval. However, Hexarelin is noted for inducing rapid receptor desensitization (tachyphylaxis) in long-term models, which limits its utility for chronic administration. Research on Hexarelin explores its potential benefits for enhancing muscle growth, improving recovery, aiding fat loss, and anti-aging applications, while it stimulates GH release without increasing appetite—a distinguishing feature compared to other GHS compounds. This GHS-R1a agonist mechanism positions Hexarelin as a critical tool compound for investigating GH-axis biology, growth hormone secretion research, anti-aging mechanisms, muscle growth pathways, fat metabolism studies, recovery enhancement, and neuroendocrine regulation in preclinical models, offering potential therapeutic insights for metabolic and endocrine disorders.

Handling & Storage Guidelines

  • Long-Term Storage: Keep lyophilized peptide sealed in original vial, protected from light and moisture; store at -20°C (-4°F) or below for optimal long-term stability (up to 3 years); stable at room temperature for several weeks; short-term storage at 2-8°C (39°F) suffices for immediate use within weeks

  • Solubility: Reconstitute with Bacteriostatic Water (2 mL recommended for 5mg vial → 0.025 mg/mL or 2.5 mg/100 mL concentration); soluble in sterile water, saline, or bacteriostatic water; swirl gently — do not vortex; avoid vigorous agitation during dissolution; avoid repeated freeze-thaw cycles; after reconstitution, store at 2-8°C under refrigeration, use within 3-4 weeks; for long-term storage of reconstituted peptide, aliquot and store at -20°C; add carrier protein (0.1% HSA or BSA) for extended stability

  • Appearance: Lyophilized white to off-white powder; reconstituted solution is clear and colorless; vials arrive at approximately 104% of labeled amount for research accuracy; peptide is hygroscopic—weigh under dry conditions

Global Logistics & Order Fulfillment

We proudly support scientific advancement across all 50 U.S. states and throughout Europe. Customers can seamlessly toggle their preferred currency between USD and EUR using the currency switcher located on the left-hand side of our website. All shipments are securely packaged to withstand international transit without compromising structural or chemical stability.

Laboratory Use Only Disclaimer

This material is sold strictly for laboratory research and development use only. It is not approved for human consumption, nor for medical, veterinary, or household applications. All purchases are governed by our standard Terms & Conditions. Please review them carefully before placing your order.

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