AC-262,536 – Solution, 300mg (10mg/mL)

AC-262,536 – Solution, 300mg (10mg/mL)

This premium, laboratory-grade research compound delivers ultra-pure AC-262,536 solution at 10mg/mL concentration in PEG400 vehicle, representing the highest standard for modern scientific investigations into selective androgen receptor modulation and tissue-specific anabolic signaling mechanisms. The ready-to-use solution format eliminates preparation time and ensures precise dosing accuracy for in vivo animal studies, eliminating solubility variability and providing investigators with a validated vehicle system ideal for analytical testing, pharmacokinetic modeling, and in vivo preclinical research applications where precise SARM administration is critical for studying beneficial anabolic effects without prostatic androgenic side effects.

All shipments to the 50 United States are fulfilled directly from primary U.S. production facilities, ensuring 2-5 business day delivery nationwide. International orders to the United Kingdom and continental Europe are processed through our dedicated United Kingdom shipping hub, which streamlines customs clearance and reduces transit times across all European countries. This dual-hub logistics infrastructure guarantees seamless, compliant delivery while maintaining chemical integrity throughout transit.

• Public third-party lab reports with unique lot-coding ensure absolute transparency for every batch sold

• Formulation contains zero adulterants, excipients, flow agents, or contaminants—pure AC-262,536 in PEG400 only

• Strategic over-fill compensates for solution adhesion loss, guaranteeing minimum 30mL (300mg) recoverable volume

• Amber glass vial features UV-resistant construction and tamper-proof seal for transit safety

Technical Specifications & Chemical Profile

Research Applications & Storage Protocols

Selective Androgen Receptor Activation & In Vivo Dosing Profiling

AC-262,536 functions as a potent and highly selective androgen receptor agonist with a K_i of 5.01 nM and EC50 of 1.58 nM in cell-based functional assays, exhibiting partial agonist activity relative to natural testosterone while demonstrating remarkable tissue selectivity. In castrated male rat models, AC-262,536 (3, 10, and 30 mg/kg oral dosing) significantly reduces plasma luteinizing hormone levels and increases levator ani muscle weight—a validated marker of anabolic activity—while producing minimal androgenic effects on prostate and seminal vesicle weights, confirming its SARM profile. The ready-to-use solution format (10mg/mL in PEG400) enables precise oral or injectable administration for in vivo studies with recommended animal dosage of 10 mg/kg, eliminating solubility variability and ensuring accurate dosing in chronic studies. A 2-week chronic study demonstrated AC-262,536 significantly improves anabolic parameters, particularly stimulating levator ani growth and suppressing elevated LH levels, without the prostatic hypertrophy associated with testosterone. This tissue-selective mechanism positions AC-262,536 solution as a critical tool compound for investigating sarcopenia mechanisms, osteoporosis treatment pathways, Alzheimer’s disease research, breast cancer models, and muscle wasting conditions in preclinical in vivo studies, offering potential therapeutic benefits without traditional androgen side effects.

Handling & Storage Guidelines

• Long-Term Storage: Store at room temperature (15-25°C) in airtight conditions; protect from light and moisture; solution remains stable for 12 months from manufacture date when stored properly

• Solubility: Pre-dissolved in PEG400 vehicle; soluble in DMSO (50 mg/mL); solution ready for direct use in oral gavage or injection formulations

• Appearance: Clear liquid solution in PEG400 vehicle; organoleptic profile: clear, colorless to pale yellow liquid

Global Logistics & Order Fulfillment

We proudly support scientific advancement across all 50 U.S. states and throughout Europe. Customers can seamlessly toggle their preferred currency between USD and EUR using the currency switcher located on the left-hand side of our website. All shipments are securely packaged to withstand international transit without compromising structural or chemical stability.

Laboratory Use Only Disclaimer

This material is sold strictly for laboratory research and development use only. It is not approved for human consumption, nor for medical, veterinary, or household applications. All purchases are governed by our standard Terms & Conditions. Please review them carefully before placing your order.