RAD140 (Testolone) – Powder, 1g

$69.99

  • RAD140 (Testolone) – Powder, 1g is ultra-pure, analytical-grade selective androgen receptor modulator (SARM) with ≥98% purity, designed for in vitro/in vivo metabolic research and analytical testing. This lyophilized material functions as an orally bioavailable, nonsteroidal SARM that binds to the androgen receptor with a Ki value of 7 nM, demonstrating high affinity and specificity for androgen receptors (ARs) with tissue-selective activity, interacting with androgenic signaling pathways while minimizing off-target interactions in prostate, skin, and sebaceous glands, making it invaluable for investigators studying muscle wasting prevention, breast cancer treatment (particularly androgen/estrogen receptor-positive breast cancer), lean body mass preservation, bone mineral density enhancement, sarcopenia reversal, cancer cachexia, athletic performance enhancement, and tissue-selective AR signaling pathways. RAD140 inhibits the growth of androgen/estrogen receptor-positive breast cancer models with a distinct mechanism of action and mimics the activity of testosterone in the body without steroidal structure. The compound is currently under development by Radius Health, Inc. (RDUS) for the treatment of conditions such as muscle wasting and breast cancer. Available for fast, compliant shipping to all U.S. states and European countries via dedicated logistics hubs.

    • Third-party certified lot coding with publicly available COA (Certificate of Analysis) for absolute purity transparency

    • Formulation completely free of flow agents, excipients, and adulterants to ensure 100% pure RAD140

    • Precision over-weighed by 5-10% inside vessel to compensate for natural adhesion loss during laboratory powder transfer

    • UV-resistant PET single-wall jar with tamper-proof seal engineered for transit safety and chemical stability

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Description

RAD140 (Testolone) – Powder, 1g

This premium, laboratory-grade research compound delivers ultra-pure raw RAD140 (Testolone) powder at ≥98% purity, representing the highest standard for modern scientific investigations into selective androgen receptor modulation and potent anabolic signaling mechanisms in muscle and bone. The lyophilized crystalline powder form provides investigators with a single-compound reference standard ideal for analytical testing, in vitro cell culture modeling of AR-mediated pathways, and in vivo preclinical research applications where precise RAD140 administration is critical for studying muscle wasting prevention, breast cancer treatment, and tissue-selective androgenic effects.

RAD140 was discovered by Radius Health, a pharmaceutical company that filed a patent for it in 2007, designed with the goal to capture the power of androgenic activity for skeletal muscle and bone, while cutting back on the unwanted side effects common with traditional androgens. As a potent SARM, RAD140 showed potential as a therapeutic agent in combating muscle wasting diseases, osteoporosis, and other conditions. RAD140 operates with laser-like focus, zoning in on androgen receptors in skeletal muscle and bone tissue to deliver its anabolic effects. It works by attaching onto the androgen receptor, triggering a conformational shift that paves the way for selective gene transcription.

All shipments to the 50 United States are fulfilled directly from primary U.S. production facilities, ensuring 2-5 business day delivery nationwide. International orders to the United Kingdom and continental Europe are processed through our dedicated United Kingdom shipping hub, which streamlines customs clearance and reduces transit times across all European countries. This dual-hub logistics infrastructure guarantees seamless, compliant delivery while maintaining chemical integrity throughout transit.

  • Public third-party lab reports with unique lot-coding ensure absolute transparency for every batch sold

  • Formulation contains zero flow agents, excipients, or adulterants—pure RAD140 only

  • Strategic over-weighing compensates for powder adhesion loss, guaranteeing minimum 1g recoverable material

  • PET single-wall jar features UV-resistant construction and tamper-proof seal for transit safety


Technical Specifications & Chemical Profile

Chemical Property Specification Data
Product Name RAD140 (Testolone) – Powder, 1g
Common Synonyms Testolone, Vosilasarm, RAD 140, EP0062, RAD-140, Testalone, Selective Androgen Receptor Modulator, SARM
CAS Number 1182367-47-0
Molecular Formula C₂₀H₁₆ClN₅O₂
Molar Mass 393.83 g/mol
Exact Mass 393.0993
IUPAC Name 2-chloro-4-{[(1R,2S)-1-[5-(4-cyanophenyl)-1,3,4-oxadiazol-2-yl]-2-hydroxypropyl]amino}-3-methylbenzonitrile
Primary Target Mechanism Orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM); binds to androgen receptor with Ki = 7 nM ; high affinity and specificity for androgen receptors (ARs); tissue-selective activity; interacts with androgenic signaling pathways while minimizing off-target interactions in prostate, skin, and sebaceous glands; mimics activity of testosterone in the body; inhibits growth of androgen/estrogen receptor-positive breast cancer models with distinct mechanism of action ; muscle wasting prevention; breast cancer treatment (androgen/estrogen receptor-positive); lean body mass preservation; bone mineral density enhancement; sarcopenia reversal; cancer cachexia; athletic performance enhancement; improves athletic performance and muscle strength; tissue-selective AR activation; investigational new drug; under development by Radius Health, Inc. (RDUS); banned in sport; on World Anti-Doping Agency (WADA) Prohibited List; banned by National Collegiate Athletic Association (NCAA); not legally allowed in dietary supplements in US; possibly unsafe; reports of heart attack and liver injury after use; liver disease contraindication; pregnancy and breast-feeding contraindication; unknown long-term safety risk; elemental analysis: C, 61.00; H, 4.10; Cl, 9.00; N, 17.78; O, 8.12
Physical Form Off-white fine powder (lyophilized solid)
Solubility Soluble in Ethanol, PEG400
Storage Room temperature ; store in a cool dry place ; minimize open air exposure ; refrigeration recommended for long-term storage
Specification ≥98% purity (HPLC verified)

Research Applications & Storage Protocols

Potent SARM-Mediated AR Agonism & Muscle/Breast Cancer Profiling

RAD140 (Testolone, Vosilasarm, EP0062) functions as an orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM) that is widely examined in preclinical research models. The compound is a type of chemical known as a selective androgen receptor modulator (SARM) that mimics the activity of testosterone in the body, providing testosterone-like effects without steroidal structure. RAD140 is designed to exhibit high affinity and specificity for androgen receptors (ARs) and is known for its tissue-selective activity, interacting with androgenic signaling pathways while minimizing off-target interactions, demonstrating superior selectivity compared to conventional androgens. It is an investigational selective androgen receptor modulator (SARM) for the treatment of conditions such as muscle wasting and breast cancer, currently under development by Radius Health, Inc. (RDUS), confirming its therapeutic development status. RAD140 Inhibits the Growth of Androgen/Estrogen Receptor Positive Breast Cancer Models with a Distinct Mechanism of Action, demonstrating unique anticancer properties beyond muscle-building effects. Due to its ability to bind to androgen receptors, the SARM has been shown to mimic the action of testosterone, providing comprehensive androgenic effects. People use testolone to improve athletic performance and muscle strength, for breast cancer, and for other purposes, demonstrating its broad research applications. This potent SARM mechanism positions RAD140 as a critical tool compound for investigating muscle wasting prevention research, breast cancer treatment models (particularly androgen/estrogen receptor-positive), lean body mass preservation studies, bone mineral density enhancement pathways, sarcopenia reversal mechanisms, cancer cachexia treatment, athletic performance enhancement, and tissue-selective androgen receptor signaling in preclinical models, offering potential therapeutic insights superior to testosterone with minimized androgenic side effects. Testolone is banned by the World Anti-Doping Agency (WADA) and the National Collegiate Athletic Association (NCAA), and there have been reports of heart attack and liver injury after use, confirming significant safety concerns for human use.

Handling & Storage Guidelines

  • Long-Term Storage: Store at room temperature in a cool, dry place away from direct light; minimize open air exposure; keep tightly sealed. Refrigeration recommended for long-term storage. PET single-wall jar provides UV resistance to minimize degradation; shelf life 36 months when stored properly

  • Solubility: Soluble in Ethanol and PEG400; prepare fresh solutions immediately before use; aqueous solutions have limited solubility; stock solutions should be prepared fresh or aliquoted and frozen for long-term storage

  • Appearance: Off-white fine powder; powder weighed out to 1.006g for 1g product (spot on accuracy); res

Global Logistics & Order Fulfillment

We proudly support scientific advancement across all 50 U.S. states and throughout Europe. Customers can seamlessly toggle their preferred currency between USD and EUR using the currency switcher located on the left-hand side of our website. All shipments are securely packaged to withstand international transit without compromising structural or chemical stability.

Laboratory Use Only Disclaimer

This material is sold strictly for laboratory research and development use only. It is not approved for human consumption, nor for medical, veterinary, or household applications. All purchases are governed by our standard Terms & Conditions. Please review them carefully before placing your order.

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