RAD140 (Testolone) – Solution, 300mg (10mg/mL)

$49.99

  • RAD140 (Testolone) – Solution, 300mg (10mg/mL) is ultra-pure, analytical-grade selective androgen receptor modulator (SARM) solution with ≥99% purity RAD140 dissolved in 99% PEG400 vehicle, designed for in vitro/in vivo metabolic research and analytical testing. This ready-to-use solution provides 10mg/mL concentration containing 300mg total RAD140 (30mL volume), functioning as an orally bioavailable, nonsteroidal SARM that binds to the androgen receptor with a Ki value of 7 nM, demonstrating high affinity and specificity for androgen receptors (ARs) with tissue-selective activity, interacting with androgenic signaling pathways while minimizing off-target interactions in prostate, skin, and sebaceous glands, making it invaluable for investigators studying muscle wasting prevention, breast cancer treatment (particularly androgen/estrogen receptor-positive breast cancer), lean body mass preservation, bone mineral density enhancement, sarcopenia reversal, cancer cachexia, athletic performance enhancement, and tissue-selective AR signaling pathways. RAD140 inhibits the growth of androgen/estrogen receptor-positive breast cancer models with a distinct mechanism of action and mimics the activity of testosterone in the body. The compound induces partial antagonist activity in seminal vesicle and prostate at 0.3-1 mg/kg, demonstrating tissue selectivity. Available for fast, compliant shipping to all U.S. states and European countries via dedicated logistics hubs.

    • Third-party certified lot coding with publicly available COA (Certificate of Analysis) for absolute purity transparency

    • Formulation: 99% PEG400 vehicle with 1% RAD140 (>99% purity) – induction sealed and batch coded

    • Precision over-filled by 5-10% inside vessel to compensate for natural solution adhesion loss during laboratory transfer

    • UV-resistant amber glass bottle with tamper-proof induction seal engineered for transit safety and chemical stability

      RAD140 (Testolone) – Solution, 300mg (10mg/mL) is ultra-pure, analytical-grade selective androgen receptor modulator (SARM) solution with ≥99% purity RAD140 dissolved in 99% PEG400 vehicle, designed for in vitro/in vivo metabolic research and analytical testing. This ready-to-use solution provides 10mg/mL concentration containing 300mg total RAD140 (30mL volume), functioning as an orally bioavailable, nonsteroidal SARM that binds to the androgen receptor with a Ki value of 7 nM, demonstrating high affinity and specificity for androgen receptors (ARs) with tissue-selective activity, interacting with androgenic signaling pathways while minimizing off-target interactions in prostate, skin, and sebaceous glands, making it invaluable for investigators studying muscle wasting prevention, breast cancer treatment (particularly androgen/estrogen receptor-positive breast cancer), lean body mass preservation, bone mineral density enhancement, sarcopenia reversal, cancer cachexia, athletic performance enhancement, and tissue-selective AR signaling pathways. RAD140 inhibits the growth of androgen/estrogen receptor-positive breast cancer models with a distinct mechanism of action and mimics the activity of testosterone in the body. The compound induces partial antagonist activity in seminal vesicle and prostate at 0.3-1 mg/kg, demonstrating tissue selectivity. Available for fast, compliant shipping to all U.S. states and European countries via dedicated logistics hubs.

      • Third-party certified lot coding with publicly available COA (Certificate of Analysis) for absolute purity transparency

      • Formulation: 99% PEG400 vehicle with 1% RAD140 (>99% purity) – induction sealed and batch coded

      • Precision over-filled by 5-10% inside vessel to compensate for natural solution adhesion loss during laboratory transfer

      • UV-resistant amber glass bottle with tamper-proof induction seal engineered for transit safety and chemical stability

Category:
Description

RAD140 (Testolone) – Solution, 300mg (10mg/mL)

This premium, laboratory-grade research compound delivers ultra-pure RAD140 (Testolone) solution at 10mg/mL concentration in optimized PEG400 vehicle, representing the highest standard for modern scientific investigations into selective androgen receptor modulation and potent anabolic signaling mechanisms in muscle and bone. The ready-to-use solution format eliminates preparation time and ensures precise dosing accuracy for in vivo animal studies, eliminating solubility variability and providing investigators with a validated vehicle system ideal for analytical testing, pharmacokinetic modeling, and in vivo preclinical research applications where precise RAD140 administration is critical for studying muscle wasting prevention, breast cancer treatment, and tissue-selective androgenic effects.

RAD140 solution utilizes 99% PEG400 as the solvent vehicle, which provides excellent solubility and bioavailability for oral and injectable research applications. The induction-sealed, batch-coded bottles ensure product integrity and traceability throughout the supply chain.

All shipments to the 50 United States are fulfilled directly from primary U.S. production facilities, ensuring 2-5 business day delivery nationwide. International orders to the United Kingdom and continental Europe are processed through our dedicated United Kingdom shipping hub, which streamlines customs clearance and reduces transit times across all European countries. This dual-hub logistics infrastructure guarantees seamless, compliant delivery while maintaining chemical integrity throughout transit.

  • Public third-party lab reports with unique lot-coding ensure absolute transparency for every batch sold

  • Formulation contains 99% PEG400 with 1% RAD140 (>99% purity) – induction sealed for security

  • Strategic over-fill compensates for solution adhesion loss, guaranteeing minimum 30mL (300mg) recoverable volume

  • Amber glass bottle features UV-resistant construction and tamper-proof induction seal for transit safety


Technical Specifications & Chemical Profile

Chemical Property Specification Data
Product Name RAD140 (Testolone) – Solution, 300mg (10mg/mL)
Common Synonyms Testolone, Vosilasarm, RAD 140, EP0062, RAD-140, Testalone, Selective Androgen Receptor Modulator, SARM, RAD140 Liquid
CAS Number 1182367-47-0
Molecular Formula C₂₀H₁₆ClN₅O₂
Molar Mass 393.83 g/mol
IUPAC Name 2-chloro-4-{[(1R,2S)-1-[5-(4-cyanophenyl)-1,3,4-oxadiazol-2-yl]-2-hydroxypropyl]amino}-3-methylbenzonitrile
Primary Target Mechanism Orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM); binds to androgen receptor with Ki = 7 nM ; high affinity and specificity for androgen receptors (ARs); tissue-selective activity; interacts with androgenic signaling pathways while minimizing off-target interactions in prostate, skin, and sebaceous glands; mimics activity of testosterone in the body; inhibits growth of androgen/estrogen receptor-positive breast cancer models with distinct mechanism of action ; partial antagonist activity in seminal vesicle and prostate at 0.3-1 mg/kg ; muscle wasting prevention; breast cancer treatment (androgen/estrogen receptor-positive); lean body mass preservation; bone mineral density enhancement; sarcopenia reversal; cancer cachexia; athletic performance enhancement; improves athletic performance and muscle strength; tissue-selective AR activation; investigational new drug; under development by Radius Health, Inc. (RDUS); banned in sport; on World Anti-Doping Agency (WADA) Prohibited List; banned by National Collegiate Athletic Association (NCAA); not legally allowed in dietary supplements in US; possibly unsafe; reports of heart attack and liver injury after use; liver disease contraindication; pregnancy and breast-feeding contraindication; unknown long-term safety risk
Physical Form Clear liquid solution (10mg/mL ±5%); 30mL total volume containing 300mg RAD140 in 99% PEG400 vehicle
Composition 99% PEG400, 1% RAD140 (>99% purity)
Concentration 1% (10mg/mL)
Application Selective Androgen Receptor Modulator

Research Applications & Storage Protocols

Potent SARM-Mediated AR Agonism & Muscle/Breast Cancer Profiling

RAD140 (Testolone, Vosilasarm, EP0062) functions as an orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM) that shows potent anabolic activity in preclinical studies. The compound is a novel, potent, orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM) that is being researched for the treatment of diseases like breast cancer and muscle atrophy. RAD140 binds to the androgen receptor with a Ki value of 7 nM, demonstrating exceptional potency for androgen receptor binding. It is designed to exhibit high affinity and specificity for androgen receptors (ARs) and is known for its tissue-selective activity, interacting with androgenic signaling pathways while minimizing off-target interactions, demonstrating superior selectivity compared to conventional androgens. At 0.3-1 mg/kg, RAD140 demonstrates partial antagonist activity in seminal vesicle and prostate, confirming tissue selectivity by acting as antagonist in prostate tissue while agonist in muscle/bone. RAD140 Inhibits the Growth of Androgen/Estrogen Receptor Positive Breast Cancer Models with a Distinct Mechanism of Action, demonstrating unique anticancer properties beyond muscle-building effects. Selective androgen receptor modulator RAD140 inhibits the growth of androgen/estrogen receptor-positive breast cancer models with a distinct mechanism of action, confirming its dual therapeutic potential for muscle wasting and breast cancer. Due to its ability to bind to androgen receptors, the SARM has been shown to mimic the action of testosterone, providing comprehensive androgenic effects. Testolone encourages an anabolic response through targeting and binding to the exclusive androgen receptors in muscles and bones, demonstrating tissue-selective targeting. RAD140 stimulates anabolism through aiming, connecting, and activating androgen receptors; however, unlike anabolic steroids, this binding tends to be restricted to the AR present in muscles and bones. Basically, it strengthens the body’s capacity to burn fats for the production of energy against the use of muscles; it destroys the fat and calorie reservoirs and protects the muscles from unnecessary wasting. This potent SARM mechanism positions RAD140 solution as a critical tool compound for investigating muscle wasting prevention research, breast cancer treatment models (particularly androgen/estrogen receptor-positive), lean body mass preservation studies, bone mineral density enhancement pathways, sarcopenia reversal mechanisms, cancer cachexia treatment, athletic performance enhancement, and tissue-selective androgen receptor signaling in preclinical models, offering potential therapeutic insights superior to testosterone with minimized androgenic side effects. Testolone is banned by the World Anti-Doping Agency (WADA) and the National Collegiate Athletic Association (NCAA), and there have been reports of heart attack and liver injury after use, confirming significant safety concerns for human use.

Handling & Storage Guidelines

  • Long-Term Storage: Minimize open air exposure; store in a cool, dry place at room temperature. Keep tightly sealed; induction sealed bottles ensure product integrity; protect from direct sunlight; amber glass bottle provides UV resistance; shelf life 24-36 months when stored properly

  • Solubility: Pre-dissolved in 99% PEG400 vehicle – ready for direct use; RAD140 is soluble in PEG400; solution is clear and stable; shake/agitate bottle before each administration for consistency

  • Appearance: Clear liquid solution; 30mL volume containing 300mg total RAD140 at 10mg/mL concentration in PEG400; <5% concentration variance for consistency; induction sealed and batch coded

Global Logistics & Order Fulfillment

We proudly support scientific advancement across all 50 U.S. states and throughout Europe. Customers can seamlessly toggle their preferred currency between USD and EUR using the currency switcher located on the left-hand side of our website. All shipments are securely packaged to withstand international transit without compromising structural or chemical stability.

Laboratory Use Only Disclaimer

This material is sold strictly for laboratory research and development use only. It is not approved for human consumption, nor for medical, veterinary, or household applications. All purchases are governed by our standard Terms & Conditions. Please review them carefully before placing your order.

Additional information
pa_feature

Discountinued

pa_form

Liquids

pa_types

SARMs

Reviews (0)

Reviews

There are no reviews yet.

Be the first to review “RAD140 (Testolone) – Solution, 300mg (10mg/mL)”